China Supplier Sell Powder CAS: 60142-96-3 Gabapentin ine Safe Delivery
Kushandisa kweGabapentin
Gabapentin(Neurontin) mushonga wemishonga, kunyanya GABA analog.Yakagadzirirwa kurapa pfari, uye iye zvino inoshandiswawo kugadzirisa kurwadziwa kweuropathic.IC50 Value: 140 nM (α2δ subunit ye calcium channel) [1]Target: Calcium Channelin vitro: Gabapentin, baclofen uye CGP 44532 zvose zvakaderedza magetsi akakurudzirwa. kuburitswa kwe [3H] glutamic acid (IC50 = 20 microM, 0.8 microM uye 2 microM, zvichiteerana).Gabapentin yakanga isina simba pakusunungurwa kwe [3H] GABA, nepo baclofen (IC50 = 8 microM) uye CGP 44532 (IC50 = 1 microM) inhibited [3H] GABA kusunungurwa [2].Kudzivirirwa kukuru kwe calcium currents ne gabapentin kwakaonekwa mu pyramidal neocortical cells (kusvika ku34%).Zvinonyanya kukosha, iyo gabapentin-mediated inhibition ye calcium currents yakazara pazvishoma zvishoma (zvakapoteredza 10 microM), zvishoma neocortical neurons (IC50 inenge 4 microM) [3].in vivo: Gabapentin yakabudisa anti-allodynic effect pamusoro pe7- nguva yezuva, kuderedza kutaura kwepro-inflammatory cytokines asi kuwedzera kutaura kweIL-10 (TNF-α, 316.0 ± 69.7 pg/mL vs 88.8 ± 24.4 pg/mL; IL-1β, 1,212.9 ± 104.5 vs 577.7. /mL; IL-6, 254.0 ± 64.8 pg/mL vs 125.5 ± 44.1 pg/mL; IL-10, 532.1 ± 78.7 pg/mL vs 918.9 ± 63.1 pg/mL).Kudzvinyirira kwegabapentin pakutaura kwepro-inflammatory cytokine kwakavharwa zvishoma ne-anti-IL-10 antibody [4]. Toxicity: Hapana zviratidzo zvitsva zvekuchengetedza kana zviitiko zvakashata zvine chokuita neGEn exposure zvakaonekwa [5] .Clinical trial: N /A
Common Name | Gabapentin | ||
---|---|---|---|
Nhamba yeCAS | 60142-96-3 | Molecular Weight | 171.237 |
Density | 1.1±0.1 g/cm3 | Boiling Point | 314.4±15.0 °C pa760 mmHg |
Molecular Formula | C9H17NO2 | Melting Point | 162°C |
Chemical & Physical Properties
Density | 1.1±0.1 g/cm3 |
---|---|
Boiling Point | 314.4±15.0 °C pa760 mmHg |
Melting Point | 162°C |
Molecular Formula | C9H17NO2 |
Molecular Weight | 171.237 |
Flash Point | 144.0±20.4 °C |
Misa chaiyo | 171.125931 |
PSA | 63.32000 |
LogP | 1.19 |
Vapor Pressure | 0.0±1.4 mmHg pa25°C |
Index yeRefraction | 1.489 |
Kuchengetedza mamiriro | Kupisa pa +4°C |
Kunyungudika kwemvura | H2O: 10 mg/mL |
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